Phortress & PMX 610 Bibliographies

Use of the COMPARE Algorithm to Guide Mechanistic Studies on Novel Antitumor Agents – a Tale of Two Benzothiazoles. Stevens MFG, Wells G, Bradshaw TD, Westwell AD and Holbeck SL. Proc. Am. Assoc. Cancer Res. 2002, 43, #4731.

Antitumor Benzothiazoles. 14. The Synthesis and In Vitro Biological Properties of Fluorinated 2-(4-Aminophenyl)benzothiazoles. Hutchinson I, Chua M-S, Browne H, Trapani V, Fichtner I, Bradshaw TD, Westwell AD and Stevens MFG. J. Med. Chem., 2001, 44, 1446-1455.

The discovery of the potent and selective antitumor agent 2-(4-amino-3-methylphenyl)benzothiazole (DF 203) and related compounds. Bradshaw TD, Stevens MFG and Westwell AD. Current Medicinal Chemistry, 2001, 8, 203-210.

Antitumor benzothiazoles. 14. The synthesis and in vitro biological properties of fluorinated 2-(4-aminophenyl)benzothiazoles. Hutchinson I, Chua M-S, Browne HL, Trapani V, Bradshaw TD, Westwell AD and Stevens MFG. J. Medicinal Chemistry, 2001, 44, 1446-1455.

Mechanistic Studies and Evaluation of Clinical Markers for Phortress, a New Agent for Clinical Trials. Bradshaw TD, Browne HL, Hutchinson I, Laughton CA, Leong CO, O’Brien S, Stevens MFG, Trapani V and Westwell AD. Brit. J. Cancer 2001, 85 (Suppl. 1), P272.

Radiolabelling of the Potential Anti-Cancer Agent, 5-Fluoro-2-(4-amino-3-methylphenyl)benzothiazole (5F203) with Fluorine-18. Brown GD, Wilson HK, Westwell AD, Hutchinson I, Stevens MFG, Price PM, Aboagye E, Luthra SK and Brady F J. Labelled Cpds. and Radiopharmaceuticals 2001, 44 (Suppl. 1), S374-S375.

Induction of CYP1A1 by 2-(4-Aminophenyl)benzothiazoles Leads to DNA Adducts in Sensitive Tumor Cells. Stevens MFG, Heydon RT, Martin EA, Farmer PB, Bradshaw TD, Hutchinson I, Westwell AD, Browne HL and Trapani V. Proc. Am. Assoc. Cancer Res., 2001, 42, 1754.

Antitumour Benzothiazoles. Part 15. The synthesis and physico-chemical properties of 2-(4-aminophenyl)benzothiazole sulfamate salt derivatives. Shi D-F, Bradshaw TD, Chua M-S, Westwell AD and Stevens MFG. Bioorg. and Med. Chem. Lett., 2001, 11, 1093-1095.

Antitumour benzothiazoles. Part 10: The synthesis and antitumour activity of benzothiazole substituted quinol derivatives. Wells G, Bradshaw TD, Diana P, Seaton A, Shi D-F, Westwell AD and Stevens MFG. Bioorg. and Med. Chem. Lett., 2000, 10, 513-515.

Mechanisms of acquired resistance to 2-(4-aminophenyl)benzothiazole (CJM 126, NSC 34445). Bradshaw TD, Chua M-S, Orr S, Matthews CS and Stevens MFG. Brit. J. Cancer, 2000, 83, 270-277.